Search results for "cholinergic excitatory nerve"

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Functional evidence for GABA as modulator of the contractility of the longitudinal muscle in mouse duodenum: Role of GABAA and GABAC receptors

2007

We investigated, in vitro, the effects of gamma-aminobutyric acid (GABA) on the spontaneous mechanical activity of the longitudinal smooth muscle in mouse duodenum. GABA induced an excitatory effect, consisting in an increase in the basal tone, which was antagonized by the GABA(A)-receptor antagonist, bicuculline, potentiated by (1,2,5,6-Tetrahydropyridin-4-yl)methylphosphinic acid hydrate (TPMPA), a GABA(C)-receptor antagonist and it was not affected by phaclofen, a GABA(B)-receptor antagonist. Muscimol, GABA(A) receptor agonist, induced a contractile effect markedly reduced by bicuculline, tetrodotoxin (TTX), hexamethonium and atropine. Cis-4-aminocrotonic acid (CACA), a specific GABA(C) …

GABA receptorsAgonistmedicine.medical_specialtyDuodenumPyridinesmedicine.drug_classIn Vitro TechniquesBicucullineInhibitory postsynaptic potentialSettore BIO/09 - FisiologiaGABAA-rho receptorGABA AntagonistsMiceGABACellular and Molecular Neurosciencechemistry.chemical_compoundPhaclofenReceptors GABAInternal medicineIntestinal motilitymedicineAnimalsDrug InteractionsGABA Agonistsgamma-Aminobutyric AcidPharmacologyDose-Response Relationship DrugMuscimolGABAA receptorCytarabineMuscle SmoothBicucullinePhosphinic AcidsMice Inbred C57BLEndocrinologyReceptors GABA-Bnervous systemchemistryMuscimolCholinergic excitatory nerveNANC inhibitory nerveHexamethoniumMouse duodenumMuscle Contractionmedicine.drugNeuropharmacology
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Functional evidence for different roles of GABAA and GABAB receptors in modulating mouse gastric tone

2010

Abstract The aims of the present study were to investigate, using mouse whole stomach in vitro , the effects of γ-aminobutyric acid (GABA) and GABA receptor agonists on the spontaneous gastric tone, to examine the subtypes of GABA receptors involved in the responses and to determine the possible site(s) of action. GABA induced gastric relaxation, which was antagonized by the GABA A -receptor antagonist, bicuculline, potentiated by phaclofen, GABA B -receptor antagonist, but not affected by 1,2,5,6-Tetrahydropyridin-4-yl methylphosphinic acid hydrate (TPMPA), GABA C -receptor antagonist. Muscimol, GABA A -receptor agonist, mimicked GABA effects inducing relaxation, which was significantly re…

Malemedicine.medical_specialtymedicine.drug_classMuscle RelaxationIn Vitro TechniquesGABAB receptorApaminSettore BIO/09 - FisiologiaMicePotassium Channels Calcium-ActivatedGABACellular and Molecular Neurosciencechemistry.chemical_compoundPhaclofenReceptors GABAGABA receptorNANC inhibitory nerves.GABA receptorInternal medicinemedicineAnimalsGABA-A Receptor AgonistsGABA-A Receptor Antagonistsgamma-Aminobutyric AcidPharmacologyGABAA receptorMuscle SmoothBicucullineReceptors GABA-AReceptor antagonistMice Inbred C57BLEndocrinologyReceptors GABA-Bnervous systemMuscimolchemistryGABA-B Receptor AgonistsMuscle Tonuscholinergic excitatory nerveNitric Oxide SynthaseGABA-B Receptor Antagonistsstomachmedicine.drugNeuropharmacology
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